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Recent advances in the development of AHR antagonists in immuno-oncology.
Sun, Lijun. 2021. “Recent Advances in the Development of AHR Antagonists in Immuno-Oncology.”. RSC Medicinal Chemistry 12 (6): 902-14.
Advances in the discovery and development of selective heme-displacing IDO1 inhibitors.
Sun, Lijun. 2020. “Advances in the Discovery and Development of Selective Heme-Displacing IDO1 Inhibitors.”. Expert Opinion on Drug Discovery 15 (10): 1223-32.
Repellendus Est Minima Laborum
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Yasmine Luise Visin joined us as Research Assistant
We welcome Yasmine to join our group as Research Assistant! She will work on developing ADMET assays.
Ganetespib, a unique triazolone-containing Hsp90 inhibitor, exhibits potent antitumor activity and a superior safety profile for cancer therapy.
Ying, Weiwen, Zhenjian Du, Lijun Sun, Kevin P Foley, David A Proia, Ronald K Blackman, Dan Zhou, et al. 2012. “Ganetespib, a Unique Triazolone-Containing Hsp90 Inhibitor, Exhibits Potent Antitumor Activity and a Superior Safety Profile for Cancer Therapy.”. Molecular Cancer Therapeutics 11 (2): 475-84.
Inhibition of Wnt Signaling in Colon Cancer Cells via an Oral Drug that Facilitates TNIK Degradation.
Zhou, Kun, Jae Eun Cheong, Subrahmanian Tarakkad Krishnaji, Aram Ghalali, Haojie Fu, Lufei Sui, Catherine Alix-Panabières, et al. 2023. “Inhibition of Wnt Signaling in Colon Cancer Cells via an Oral Drug That Facilitates TNIK Degradation.”. Molecular Cancer Therapeutics 22 (1): 25-36.
Plant flavonoid inhibition of SARS-CoV-2 main protease and viral replication.
Lin, Lin, Da-Yuan Chen, Christina Scartelli, Huanzhang Xie, Glenn Merrill-Skoloff, Moua Yang, Lijun Sun, Mohsan Saeed, and Robert Flaumenhaft. 2023. “Plant Flavonoid Inhibition of SARS-CoV-2 Main Protease and Viral Replication.”. IScience 26 (9): 107602.
Topical Application of a Mast Cell Stabilizer Improves Impaired Diabetic Wound Healing.
Tellechea, Ana, Sha Bai, Seema Dangwal, Georgios Theocharidis, Masa Nagai, Steffi Koerner, Jae Eun Cheong, et al. 2020. “Topical Application of a Mast Cell Stabilizer Improves Impaired Diabetic Wound Healing.”. The Journal of Investigative Dermatology 140 (4): 901-911.e11.
Novel Reversible Fluorescent Glycan Linker for Functional Glycomics.
Wei, Mohui, Tanya R McKitrick, Akul Y Mehta, Chao Gao, Nan Jia, Alyssa M McQuillan, Jamie Heimburg-Molinaro, Lijun Sun, and Richard D Cummings. 2019. “Novel Reversible Fluorescent Glycan Linker for Functional Glycomics.”. Bioconjugate Chemistry 30 (11): 2897-2908.